Search Result "X receptor (PXR)"


Pregnane X Receptor (PXR) at the Crossroads of Human Metabolism and Disease

Journal: Current Drug Metabolism
Volume: 14 Issue: 3 Year: 2013 Page: 341-350
Author(s): Ioannis Koutsounas,Stamatios Theocharis,Efstratios Patsouris,Constantinos Giaginis

Ligand-Dependent Assembly of Pregnane X Receptor, Constitutive Androstane Receptor and Liver X Receptor Is Applicable to Identify Ligands

Journal: Drug Metabolism Letters
Volume: 4 Issue: 2 Year: 2010 Page: 88-94
Author(s): Kaoru Kobayashi, Kosuke Saito, Sachiko Takagi, Kan Chiba

Nuclear Receptors CAR and PXR in Metabolism and Elimination of Drugs

Journal: Current Pharmacogenomics
Volume: 1 Issue: 2 Year: 2003 Page: 75-85
Author(s): P. Honkakoski

Post-translational and Post-transcriptional Modifications of Pregnane X Receptor (PXR) in Regulation of the Cytochrome P450 Superfamily

Journal: Current Drug Metabolism
Volume: 14 Issue: 10 Year: 2013 Page: 1059-1069
Author(s): Tomas Smutny,Sridhar Mani,Petr Pavek

Structure and Function of the Human Nuclear Xenobiotic Receptor PXR

Journal: Current Drug Metabolism
Volume: 6 Issue: 4 Year: 2005 Page: 357-367
Author(s): V. E. Carnahan, M. R. Redinbo

New Opportunities for Pregnane X Receptor (PXR) Targeting in Drug Development. Lessons from Enantio- and Species-Specific PXR Ligands Identified from A Discovery Library of Amino Acid Analogues

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 7 Issue: 6 Year: 2007 Page: 617-625
Author(s): Peter Wipf, Haibiao Gong, Jelena M. Janjic, Song Li, Billy W. Day, Wen Xie

Research Article

Transactivation Assays that Identify Indirect and Direct Activators of Human Pregnane X Receptor (PXR, NR1I2) and Constitutive Androstane Receptor (CAR, NR1I3)

Journal: Drug Metabolism Letters
Volume: 11 Issue: 2 Year: 2017 Page: 128-137
Author(s): Marija Pinne,Elsa Ponce,Judy L. Raucy

Xenosensors CAR and PXR at Work: Impact on Statin Metabolism

Journal: Current Drug Metabolism
Volume: 12 Issue: 3 Year: 2011 Page: 300-311
Author(s): Maria Marino, Alessandra di Masi, Viviana Trezza, Valentina Pallottini, Fabio Polticelli, Paolo Ascenzi

Pregnane X Receptor and its Potential Role in Drug Resistance in Cancer Treatment

Journal: Recent Patents on Anti-Cancer Drug Discovery
Volume: 4 Issue: 1 Year: 2009 Page: 19-27
Author(s): Yakun Chen, Daotai Nie

Ligand Recognition by Drug-Activated Nuclear Receptors PXR and CAR: Structural, Site-Directed Mutagenesis and Molecular Modeling Studies

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 6 Issue: 8 Year: 2006 Page: 937-943
Author(s): Antti Poso, Paavo Honkakoski

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